Annotation Detail

Information
Associated Genes
GSTP1
Associated Variants
GSTP1 UNDEREXPRESSION
Source Database
MMMP
Description
Combined inhibition of both GSTP1 and MRP1 (ABCC1) with siRNA and sulphinpyrazone, respectively, sensitizes melanoma cells to etoposide
MMMP State
downregulated by
MMMP Molecule
GSTP1, MRP1
MMMP Modifier
GSTP1 siRNA + Sulphinpyrazone
MMMP Relationship
sensitivity to
MMMP Drug
Etoposide
MMMP Drug Alias
VP-16
MMMP Model
3
MMMP Reference
Depeille P, Br J Cancer 2005, 93:216-23
Drugs
Drug NameSensitivitySupported
EtoposideSensitivitytrue